Umukandara n'Inzira: Ubufatanye, Ubwumvikane no Gutsinda Ubwuzuzanye
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Ibicuruzwa

Teduglutide CAS:197922-42-2 Umukozi Ukora

Teduglutide (izwi kandi nka ALX-0600) ni ubwoko bwa GLP-2 aho glycine yasimbuwe na alanine ku mwanya wa 2 uvuye kuri N-terminus, bityo igatanga ubudahangarwa bwo kwangirika na DPP-4. Teduglutide ifite ubushobozi bwo gufatanya, imbaraga za agonist, n'ubushobozi bwa agonist nk'ubwa GLP-2 mu isuzuma hamwe na receptor ya GLP-2 y'imbeba. Gutanga teduglutide ku mbeba byatumye ibiro by'amara mato byiyongera cyane ndetse binatuma uburebure bwa villi y'amara bwiyongera. Teduglutide yateguwe hakoreshejwe peptide ikora mu buryo bwa solid-phase.


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Ishyirwa mu bikorwa n'ingaruka

Teduglutide ni imisemburo ya peptide ikoreshwa mu kuvura abarwayi b'abana mu gihe kirekire. Byagaragaye ko igira akamaro mu kuvura indwara z'ubwiyongere bw'umubiri n'indwara z'amara. Ni peptide imeze nka glucagon-like peptide 1 (GLP-1) ikora igihe kirekire. Byagaragaye ko uyu muti ufite ubushobozi bwo guhagarara neza mu binyabutabire, bivuze ko udacika byoroshye. Teduglutide iterwa mu mubiri ikajyanwa mu turemangingo, aho ikora receptors ku buso bw'uturemangingo. Uku gukora gutuma umwijima ukora isukari nyinshi kandi bigatuma insuline irushaho kuba nziza mu ngingo zo mu gice cy'umubiri nko mu mitsi, ibinure, n'umwijima. Yongera kandi umuvuduko w'umutima n'amaraso.

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Amakuru y'inyongera:

Imiterere C164H252N44O55S
Isuzuma 99%
Isura Ifu y'umweru kuva kuri umweru utari umweru
Nimero ya CAS 197922-42-2
Gupakira 25KG
Igihe cyo kuruhuka Imyaka 2
Ububiko Bika ahantu hakonje kandi humutse
Icyemezo ISO.

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