-
β-Nicotinamide Adenine Dinucleotide Phosphate Disodium Umunyu CAS:24292-60-2
β-Nicotinamide Adenine Dinucleotide Phosphate Disodium Umunyuni coenzyme ikwirakwira cyane mu bintu bizima, igira uruhare mu kugabanya ogisijeni. Ikora nk'umuyoboro wa electron mu bikorwa bitandukanye, ikaba ihinduka ogisijeni mu buryo bunyuranye (NADP+) ikagabanuka (NADPH).β-Nicotinamide Adenine Dinucleotide Phosphate Disodium Umunyuni ikintu kirimo aside nikotine amide adenine dinucleotide na molekile ya fosfeti bihuzwa na ester bond. Ni receptor ya hydrogène kandi ishobora gukoreshwa mu guteza imbere no guteza imbere reagents zitandukanye zo gusuzuma indwara muri vitro.
-
β-Nicotinamide Adenine Dinucleotide Umunyu wa Litiyumu (umunyu wa LADIYA NAD) CAS: 64417-72-7
β-Nicotinamide Adenine Dinucleotide Umunyu wa Lithiumni coenzyme ikomeye mu mikorere y'umubiri. Iboneka mu turemangingo twose tuzima, NAD yitwa dinucleotide kuko igizwe na nucleotide ebyiri zihujwe binyuze mu matsinda yazo ya fosifate. Nucleotide imwe irimo adenine nucleobase n'indi nicotinamide. NAD ibaho mu buryo bubiri: imiterere ya oxidized n'igabanuka, mu magambo ahinnye nka NAD+ na NADH (H isobanura hydrogen), uko bikurikirana.
-
Venlafaxine CAS: 93413-69-5
Venlafaxine ni umuti ugabanya ubukana bw'indwara zo mu bwoko bwa serotonin na norepinephrine reuptake inhibitor (SNRI). Uyu muti wakozwe bwa mbere na Wyeth muri 19Chemicalbook93 none ubu ugurishwa na Pfizer. Uyu muti wemejwe mu kuvura indwara ikomeye yo kwiheba (MDD), indwara yo guhangayika rusange (GAD), n'ihungabana rijyanye no guhangayika.
-
Umukozi ushinzwe imikorere ya Ciclopirox Ethanolamine CAS:41621-49-2
Ciclopirox ethanolamine ni umuti urwanya imiyoboro y'amaraso mu buryo bwagutse, kandi urwanya bagiteri nyinshi za Gram-positive na Gram-negative, kandi ufite ubushobozi bwo kurwanya ububyimbirwe. Ikoreshwa mu kuvura indwara z'uruhu n'inzara.
-
Desvenlafaxine Yatsinze CAS: 386750-22-7
Desvenlafaxine Succinate ni umuti ugabanya ubukana bwa serotonin na norepinephrine (SNRI) wemejwe mu kuvura indwara ikomeye yo kwiheba (MDD) muri Leta Zunze Ubumwe za Amerika mu 2008. Kugira ngo venlafaxine irusheho kugira akamaro n'umutekano, Wyeth yavumbuye kandi akora imwe mu miti ikomeye ya venlafaxine, ari yo O-desmethyl metabolite (desvenlafaxine).
-
Doxazosin Mesylate CAS: 77883-43-3 Umukozi Ukora
Doxazosin mesylate ni quinazoline compound igabanya ubukana bw'ubwoko bwa alpha1 bwa alpha adrenergic receptors. Doxazosin mesylate ni ubwoko bushya bwa quinazolone α1 receptor blocker yakozwe na Pfizer sosiyete (Leta Zunze Ubumwe za Amerika), ifite igihe kirekire cyo kumara igice cy'ubuzima, ikora ingaruka zo kwagura imiyoboro y'amaraso, kugabanya ubudahangarwa bw'imitsi no kugabanya umuvuduko w'amaraso binyuze mu kuziba receptor ya a 1. Yagiriwe inama mu mahanga nk'imiti ya mbere ivura indwara ya hypertension no kuvura indwara ya prostate.
-
L-Isoleucine CAS: 73-32-5 Umukozi Ukora
L-Isoleucine, izwi kandi nka Isoleucine, ni aside amine igizwe n'isomeri ya leucine. Ni ingenzi mu gukora hemoglobine no kugenzura urugero rw'isukari n'ingufu mu maraso. L-Isoleucine ni isomeri ya L-leucine kandi ni aside amine y'ingenzi. Ikorwa muri threonine kandi ni aside amine ikomoka ku miyoboro y'amazi.
-
Captopril CAS: 62571-86-2 Umukozi Ukora
Captopril ni yo miti igabanya umuvuduko w'amaraso mu mitsi igabanya umuvuduko w'amaraso mu mubiri (angiotensin-converting enzymes) ikoreshwa mu bushakashatsi bwinshi bwakozweho nk'umuti ugabanya umuvuduko w'amaraso mu mubiri. Ihagarika enzyme ihindura amaraso mu mubiri, igabanya ikorwa rya angiotensin II kandi ikagabanya ingaruka zayo zo kugabanya imitsi mu mitsi n'imitsi. Umuvuduko w'amaraso mu mitsi uragabanuka, bigatuma umuvuduko w'amaraso ugabanuka.
-
Candesartan CAS: 139481-59-7 Umukozi Ukora
Candesartan ni antagonist ya angiotensin II receptor I (AT1), IC50s = 1.12 na 2.86 nM kuri cortex y'inka na aorta y'urukwavu. Ibuza igabanuka rya angiotensin II riterwa na angiotensin II ry'imirongo ya aorta y'urukwavu nta ngaruka igira ku igabanuka riterwa n'ibindi bintu nka norepinephrine, KCl, serotonin, PGF2α cyangwa endothelin.
-
Candesartana Cilexetila CAS:145040-37-5
Candesartan Celexetil ni ester analog y'umurwanyi wa angiotensin II Candesartan (sc-217825). Urwango rw'iyi receptor rubuza angiotensin II gufatana, vasoconstrictor ikomeye. Ibi bigira ingaruka rusange zo kwaguka kw'imitsi no kwiyongera k'umuvuduko w'amaraso mu mitsi. Candesartan Celexetil Ester ni umurinzi wa AT1.
-
Bupropion CAS: 34911-55-2 Umukozi Ukora
Bupropion ni aromatic ketone ari yo propiophenone itwara itsinda rya tert-butylamino ku mwanya wa 2 n'isimbura chloro ku mwanya wa 3 ku mpeta ya phenyl. Ifite uruhare mu kugabanya ubudahangarwa bw'umubiri, kwanduza ibidukikije no kuba xenobiotic. Ni amino ya kabiri, ikaba igize monochlorobenzenes na aromatic ketone.
-
Bezafibrate CAS: 41859-67-0 Umukozi Ukora
Bezafibrate ni aside monocarboxylic amide iboneka mu gushonga kwemewe kw'itsinda rya karuboxy rya aside 4-chlorobenzoic hamwe n'itsinda rya amino rya aside 2-[4-(2-aminoethyl)phenoxy]-2-methylpropanoic. Benafibrate ikoreshwa mu kuvura hyperlipidemia. Ifite uruhare nk'umuti wa xenobiotic, umuti wanduza ibidukikije, umurinzi wa gero n'umuti urwanya lipemic. Ni aside monocarboxylic, ether ihumura, igice cya monochlorobenzenes na aside monocarboxylic amide. Ifitanye isano n'imikorere ya aside propionic.
