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Hygromycin B CAS: 31282-04-9
Hygromycin B ni umuti urwanya udukoko ukomoka kuri Streptomyces hygroscopicus ukunze gukoreshwa mu binyabuzima bya molekile no mu miterere y’uturemangingo. Uzwiho ubushobozi bwo kubuza poroteyine gukora binyuze mu kwivanga muri ribosome, bigatuma ugira ingaruka nziza ku bwoko butandukanye bwa bagiteri, ibihumyo, n’uturemangingo twinshi twa eukaryotic. Hygromycin B ikunze gukoreshwa nk'ikintu gitoranya mu buhanga mu by’imiterere y’uturemangingo kugira ngo hamenyekane uturemangingo twahinduwe twashyizemo uturemangingo twirwanya iyi miti.
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Imipenem anhydrous CAS: 64221-86-9
Imipenem anhydrous ni umuti urwanya udukoko twinshi ukomoka mu bwoko bwa carbapenem, uzwiho kugira ingaruka nziza ku ndwara zitandukanye za bagiteri. Ukora mu kubuza imikorere y’uturemangingo tw’uturemangingo twa bagiteri, bigatuma uba uburyo bukomeye bwo kuvura indwara zikomeye ziterwa na bagiteri zidashobora imiti myinshi. Imipenem anhydrous ikunze gukoreshwa mu buvuzi mu kuvura indwara zikomeye zo mu nda, umusonga, indwara zo mu nzira y’inkari, na sepsis bitewe nuko ikwirakwira cyane kuri bagiteri za gram-positive na gram-negative.
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Hexamidine diisethionate CAS: 659-40-5
Hexamidine diisethionate ni imvange y’ibikomoka ku ruhu ifite ubushobozi bwo kurwanya indwara ziterwa no kubyimba. Ikunze gukoreshwa mu bikoresho byo kwita ku ruhu kubera ubushobozi bwayo bwo kurwanya indwara zitandukanye z’uruhu. Iki kintu kizwiho kugira ubushobozi bwo kurwanya bagiteri no kugabanya ububyimbirwe ku ruhu, bigatuma kiba cyiza mu kuvura ibiheri, eczema, n’ibindi bibabaza uruhu. Hexamidine diisethionate ishobora gufasha mu kubungabunga uruhu rwiza irurinda kurwara kandi rudafite udukoko twangiza, bigatuma uruhu rugira isura nziza kandi ikagira ubuziranenge.
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Geldanamycin CAS: 30562-34-6
Geldanamycin ni umuti usanzwe ukomoka kuri Streptomyces hygroscopicus. Ni uwo mu bwoko bwa benzoquinone ansamycins kandi ufite ubushobozi bukomeye bwo kurwanya kanseri kuko ubuza poroteyine yo gushyuha 90 (Hsp90), poroteyine ya chaperone ikenewe cyane kugira ngo uturemangingo twa kanseri turambe. Geldanamycin yagaragaje icyizere mu bushakashatsi bwakozwe mbere yo kuvura kanseri nk'umuti ushobora kuvura ubwoko butandukanye bwa kanseri.
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Furazolidone CAS: 67-45-8
Furazolidone ni antibiyotike ikoze muri nitrofuran ifite ubushobozi bwo kurwanya indwara zandura mu buryo bwagutse. Ikunze gukoreshwa mu kuvura indwara zandura za bagiteri na protozoa haba mu buvuzi bw'amatungo no mu bantu. Furazolidone ikora mu kubuza gukura kwa bagiteri n'udukoko binyuze mu kubangamira imikorere yabyo ya metabolic. Iyi antibiyotike izwiho kugira imbaraga mu kurwanya bagiteri zitandukanye za Gram-positive na Gram-negative, ndetse na protozoa zimwe na zimwe.
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Halquinol CAS: 8067-69-4
Halquinol ni umuti w’amatungo urwanya udukoko urwanya udukoko, ukaba ufite ubushobozi bwo kurwanya udukoko duto cyane kandi tugatera indwara. Ni mu bwoko bwa 8-hydroxyquinoline, kandi ikoreshwa cyane mu matungo no mu musaruro w’inkoko mu kurwanya no gukumira indwara zo mu mara ziterwa na bagiteri na protozoa. Halquinol ifasha mu kunoza ubuzima bw’amatungo no gukora neza binyuze mu kwibasira udukoko twinshi mu nzira y’igifu.
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Genetine disulfate (G418 sulfate) CAS: 108321-42-2
Genetine disulfate, izwi kandi nka G418 sulfate, ni antibiyotike ikomeye ikomoka kuri Micromonospora rhodorangea. Iri mu bwoko bwa antibiyotike za aminoglycoside kandi ikoreshwa cyane mu bushakashatsi ku binyabuzima bya molekile nk'ikintu gihitamo sisitemu yo kwita ku turemangingo. Genetine disulfate ibuza poroteyine mu turemangingo twa prokaryotic na eukaryotic ihuza na ribosome, bigatuma igira akamaro mu guhitamo uturemangingo twahinduwe tugaragaza uturemangingo twa resistance.
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Imipenem monohydrate CAS: 74431-23-5
Imipenem monohydrate ni umuti ukomeye wa antibiyotike ukomoka mu bwoko bwa carbapenem, ugira ingaruka ku ndwara zitandukanye za bagiteri. Ikora mu kubuza imikorere y’urukuta rw’uturemangingo twa bagiteri, bigatuma igira akamaro mu kuvura indwara zikomeye ziterwa na bagiteri zidashobora imiti myinshi. Imipenem monohydrate ikoreshwa cyane mu buvuzi mu kuvura indwara zikomeye zo mu nda, umusonga, indwara zo mu nzira y’inkari, na sepsis bitewe nuko ikwirakwira cyane mu kurwanya bagiteri za gram-positive na gram-negative.
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Gramicidin CAS: 1405-97-6
Gramicidin ni antibiyotike ya peptide ikorwa na bagiteri ya Bacillus brevis. Iri mu bwoko bwa lipopeptides zikora ku buryo busanzwe kandi izwiho ubushobozi bwayo bwo kurwanya mikorobe za Gram-positive. Gramicidin ibangamira uturemangingo twa bagiteri, bigatuma ibikubiye mu turemangingo biva mu turemangingo bigahitana uturemangingo. Ikoreshwa cyane mu miti ikoreshwa mu kuvura indwara zo mu bwoko bwa peptide, cyane cyane mu bicuruzwa bivanze, mu kuvura indwara zo mu bwoko bwa virus.
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Malonamide CAS: 108-13-4
Malonamide ni ikinyabutabire gifite formula ya C3H6N2O, izwiho gukoreshwa nk'igice cy'ingenzi mu guhuza imiterere y'ibinyabuzima. Igizwe n'amatsinda abiri ya amide afatanye n'umugongo wa aside malonic. Malonamide ikunze gukoreshwa mu bushakashatsi ku miti no mu nganda zikora imiti bitewe n'uburyo ikora ibintu byinshi bitandukanye ndetse n'ubushobozi bwo gukora imiterere ikomeye ya molekile.
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H-Pyrrolo[2,3-b]pyridine,4-bromo- CAS:348640-06-2
H-Pyrrolo [2,3-b]pyridine, 4-bromo- ni imvange y’ibinyabutabire ifite formula ya molekile C9H6BrN. Iri mu cyiciro cya pyrrolopyridine cy’ibinyabutabire bya heterocyclic kandi ifite atome ya bromine iri ku mwanya wa 4. Iyi mvange izwiho imiterere yayo n’akamaro kayo mu gukora organic synthesis. H-Pyrrolo [2,3-b]pyridine, 4-bromo- ikora nk'inkingi y'agaciro mu gutegura molekile zitandukanye bitewe n'uburyo ikora neza kandi ishobora gukoreshwa.
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Methyl4-amino-2-methoxybenzoate CAS:27492-84-8
Methyl 4-amino-2-methoxybenzoate ni imvange y’ibinyabutabire ifite formula ya molekile C9H11NO3. Igizwe n’imvange y’aside benzoic yasimbuwe n’itsinda ry’amino riri ku mwanya wa 4 n’itsinda ry’aside methoxy riri ku mwanya wa 2. Iyi mvange igaragaza imiterere yihariye y’ibinyabutabire ituma igira agaciro mu buryo butandukanye bwo gukora ibintu bikomoka ku binyabuzima no mu bushakashatsi.
