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5-Bromo-2-chloro-4-(cyclopentylamino)pyrimidine CAS:733039-20-8
5-Bromo-2-chloro-4- (cyclopentylamino)pyrimidine ni ikinyabutabire cyakoreweho ubushakashatsi mu by'imiti. Gifite imiterere ya pyrimidine irimo bromo na chloro, ishobora kugira akamaro mu kuvura, ikaba igamije uburyo bwihariye bw'indwara cyangwa inzira za biyoloji mu kuvumbura imiti.
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4-[6-[[6-(1-Butoxyvinyl)-8-cyclopentyl-5-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino]pyridin-3-yl]piperazine-1-aside kaboksilike tert-butyl ester CAS:866084-31-3
4-[6-[[6-(1-Butoxyvinyl)-8-cyclopentyl-5-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino]pyridin-3-yl]piperazine-1-carboxylic acid tert-butyl ester ni ikinyabutabire cy’urusobe gifite umugongo wa piperazine ufite amatsinda mato arimo pyridine, pyrimidine, na tert-butyl ester. Imiterere yayo ishyigikira ikoreshwa rishobora gukoreshwa mu buvuzi no mu iterambere ry’imiti bitewe n’uburyo butandukanye bwo kuyikoresha mu buvuzi.
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Bortezomib CAS: 179324-69-7
Bortezomib ni umuti ukoreshwa mu kuvura indwara ya myeloma nyinshi na lymphoma ya mantle cell. Ni mu itsinda ry’imiti igabanya ubukana bwa proteasome, ikaba yibanda ku misemburo ya proteolytic mu turemangingo kugira ngo ihagarike imikorere yatwo no gutera apoptosis (urupfu rw’uturemangingo rwateguwe). Ubu buryo butuma igira ingaruka nziza ku ndwara zimwe na zimwe za kanseri aho ingirabuzimafatizo zikura mu buryo butagenzurwa.
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Methyl 2-bromomethyl-3-nitrobenzoate CAS:98475-07-1
Methyl 2-bromomethyl-3-nitrobenzoate ni imvange y'ibinyabutabire irimo itsinda rya nitro riri ku mwanya wa 3 n'itsinda rya bromomethyl riri ku mwanya wa 2 w'umugongo wa benzoate. Ikoreshwa mu guhuza ibinyabuzima nk'igikoresho cy'ikoranabuhanga, gituma habaho iyubakwa ry'uturemangingo duto dufite amatsinda yihariye y'imikorere.
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Pemetrexed disodium INT-5 CAS: 165049-28-5
Pemetrexed disodium INT-5 ni umuti uvura kanseri ugizwe n’imiti irwanya kanseri ya chimiotherapie. Ukoreshwa cyane cyane mu kuvura kanseri zitandukanye, harimo mesothelioma, kanseri y’ibihaha itari iy’uturemangingo duto, na kanseri yihariye ya metastasis.
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Pemetrexed disodium INT-4 CAS: 137281-39-1
Pemetrexed disodium INT-4 ni umuti urwanya kanseri ya kanseri ukoreshwa mu buvuzi bwa kanseri. Ukoreshwa mu kuvura kanseri zitandukanye, harimo mesothelioma, kanseri y'ibihaha itari iy'uturemangingo duto, na kanseri yihariye ya metastasis.
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Pemetrexed disodium INT-3 CAS: 155405-80-4
Pemetrexed disodium INT-3 ni umuti urwanya folate chemotherapy ukoreshwa muri kanseri. Ukoreshwa mu kuvura kanseri zitandukanye, harimo mesothelioma, kanseri y'ibihaha itari iy'uturemangingo duto, na kanseri yihariye ya metastasis.
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Ishingiro rya Terbinafine CAS: 91161-71-6
Terbinafine base ni ikintu cy’ingenzi mu miti gikoreshwa mu kuvura indwara z’ibihumyo. Ni mu bwoko bwa allylamine bw’imiti irwanya udukoko kandi izwiho kugira ingaruka nziza ku ndwara ziterwa n’udukoko two mu bwoko bwa dermatophyte, imisemburo n’ibihumyo.
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2-Chloro-4,6-dimethoxy-1,3,5-triazine CAS:3140-73-6
2-Chloro-4,6-dimethoxy-1,3,5-triazine ni imvange y’ibinyabutabire ikoreshwa nk’inkingi ikomeye mu guhuza ibinyabuzima no guhindura imiterere yabyo. Ifite imiterere ya chloro na methoxy ifatanye n’imiterere y’impeta ya triazine, bigatuma ikoreshwa mu buryo butandukanye bw’ibinyabutabire n’imiterere y’ibinyabutabire.
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2-Amino-4,5-bis (2-methoxyethoxy)benzonitrile CAS:950596-58-4
2-Amino-4,5-bis (2-methoxyethoxy)benzonitrile ni ikinyabutabire gikoreshwa mu bushakashatsi ku miti, kirangwa n'imiterere ya benzonitrile hamwe n'ibisimbura amino na methoxyethoxy, bishobora kuba ingenzi mu mikorere yihariye yo kuvura.
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(1R)-(S)-pinanediol-1-Ammonium Trifluoroacetate-3-methlbutane-1-boronate CAS:179324-87-9
(1R)-(S)-Pinanediol-1-Ammonium Trifluoroacetate-3-Methylbutane-1-Boronate ni ikinyabutabire kirangwa n'imiterere igoye irimo umugongo wa pinanediol, itsinda rya ammonium trifluoroacetate, n'imikorere ya ester ya boronate. Ikoreshwa mu guhuza ibinyabuzima nk'inkingi y'ubwubatsi bwa chiral, bigatuma habaho imvange yihariye n'ibindi bikoresho by'imiti.
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Diethyl L-glutamate hydrochloride CAS: 1118-89-4
Diethyl L-glutamate hydrochloride ni ikinyabutabire gikoreshwa cyane cyane nk'igice cy'ubuvanganzo mu bushakashatsi ku miti no mu guhuza ibinyabuzima. Kiva muri aside L-glutamic kandi kikaba ari ingenzi mu gukora imiti itandukanye n'ibindi bintu bikora ku buzima bw'umuntu.
