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Empagliflozin CAS: 864070-44-0 Umukozi Ukora

Empagliflozin ni imvange ya C-glycosyl igizwe n'ibisigazwa bya beta-glucosyl bifite itsinda rya (4-chloro-3-{4-[(3S)-tetrahydrofuran-3-yloxy]benzyl}phenyl mu kigo cy'amazi. Imvange ya sodium-glucose co-transporter 2 ikoreshwa nk'inyongera ku mirire no gukora imyitozo ngororamubiri kugira ngo yongere kugenzura glycemic ku bantu bakuru barwaye diyabete yo mu bwoko bwa 2. Ifite uruhare nk'imvange ya sodium-glucose transport protein subtype 2 kandi igabanya hypoglycemia. Ni imvange ya C-glycosyl, aromatic ether, tetrahydrofuryl ether kandi ikaba n'igice cya monochlorobenzenes.


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Empagliflozin ni umuti mushya, ukomeye kandi utoranya SGLT-2, utuma isukari igabanuka mu mubiri igenzurwa neza n’imiterere y’indwara ya metabolic mu mbeba zirwaye diyabete. Empagliflozin (izina ry’ubucuruzi Jardiance) ni umuti ugabanya isukari ya sodium glucose co-transporter-2 (SGLT-2), kandi utuma isukari mu maraso isohoka mu mpyiko ikajya mu nkari. Empagliflozin ishobora gutera umwuma no kugabanya umuvuduko w’amaraso, bigatuma abarwayi bagira isereri cyangwa gucika intege no kugabanuka k’imikorere y’impyiko. Ingaruka z’abarwayi bakuze, cyane cyane abafite ikibazo cy’imikorere y’impyiko n’imiti igabanya amaraso, zisa nkaho ari nyinshi. FDA isaba Boehring na Eli Lilly gukora inyigo enye nyuma yo kwamamaza: inyigo zuzuye z’imitsi n’umutima, inyigo z’imiti n’imiti ku bana, inyigo z’umutekano n’ubushobozi bw’abana, isuzuma ry’uburozi bw’uyu muti (cyane cyane ingaruka ku mikorere y’impyiko, imikurire n’imikurire y’amagufwa).

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Amakuru y'inyongera:

Imiterere C23H27ClO7
Isuzuma 99%
Isura Ifu y'umweru
Nimero ya CAS 864070-44-0
Gupakira 25KG
Igihe cyo kuruhuka Imyaka 2
Ububiko Bika ahantu hakonje kandi humutse
Icyemezo ISO.

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