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Ibicuruzwa

Sitagliptin Phosphate CAS: 654671-78-0 Umukozi Ukora

Fosfate ya Sitagliptinni wo muti wa mbere mushya wa dipeptidyl peptidase IV ukoreshwa na Merck mu kuvura diyabete yo mu bwoko bwa 2 utiyongera ibiro kandi umubare w’abarwaye hypoglycemia wari usa n’uwa placebo. Sitagliptin ikora mu kongera sisitemu ya incretin mu mubiri, ifasha mu kugenga isukari binyuze mu kugira ingaruka ku turemangingo twa β na α mu impyiko.


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Sitagliptin Phosphate ni umuti ugabanya glucose mu maraso wa trizolopyrazine dipeptidyl peptidase IV. Sitagliptin iherutse kwemererwa kuvura diyabete yo mu bwoko bwa II. Sitagliptin phosphate ni umuti wo mu bwoko bwa dipeptidyl peptidase Ⅳ (DDP-4) wakozwe n'ikigo cy'Abadage cya Merck, hanyuma ubanza kwemererwa n'Ikigo cy'Ibiribwa n'Imiti cya Amerika mu kuvura diyabete yo mu bwoko bwa 2, ni umuti mushya urwanya diyabete, ushobora kunoza ubushobozi bw'umubiri bwo kugabanya urugero rwinshi rwa glucose mu maraso, no kwiyongera kwa incretin mu buryo busanzwe binyuze mu kubuza imikorere y'iyi enzyme, harimo urugero rwa peptide 1 imeze nka glucagon na peptide insulinotropic ishingiye kuri glucose, bityo bigatuma pancreas yongera umusaruro wa insuline kandi igahagarika umusaruro wa glucose mu mwijima, kandi amaherezo ikagabanya ingaruka z'ubwinshi bw'glucose mu maraso.

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图片 364 (1)
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Gupakira ibicuruzwa:

8 338 (1)

Amakuru y'inyongera:

Imiterere C16H15F6N5O.H3PO4
Isuzuma 99%
Isura Ifu y'umweru kuva kuri umweru utari umweru
Nimero ya CAS 654671-78-0
Gupakira 25KG
Igihe cyo kuruhuka Imyaka 2
Ububiko Bika ahantu hakonje kandi humutse
Icyemezo ISO.

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