Umukandara n'Inzira: Ubufatanye, Ubwumvikane no Gutsinda Ubwuzuzanye
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Olmesartan Medoxomil CAS: 144689-63-4 Umukozi Ukora

Olmesartan Medoxomil, ni umuti mushya udasanzwe kandi urwanya angiotensin II yo mu bwoko bwa 1 receptor antagonist kandi urwanya cyane imikorere ya Ang.ll-induced pressor responses. Uyu muti wabujije uburyo bwo gufatana kwa [125I1]-All kuri AT1 receptors mu ruhu rw'inka, ariko nta ngaruka wagize ku gufatana kwa AT2 receptors mu ruhu rw'inka. Olmesartan medoxomil yagaragaye kandi ko igabanya umuvuduko w'amaraso neza cyane kurusha losartan na ACE inhibitor captopril ndetse na pbloker atenolol.


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Olmesartan medoxomil ni umuti urwanya angiotensin II receptor ukoreshwa mu kuvura umuvuduko ukabije w'amaraso. Olmesartan ikora mu kubuza angiotensin II gufatana na AT1 receptors mu mitsi y'amaraso. Mu kubuza gufatana aho gukora angiotensin II, olmesartan ibuza uburyo bubi bwo kugenzura isohoka rya renin. Olmesartan medoxomil ni umuti ufasha mu gukuraho metabolite ikora, olmesartan. Olmesartan ifite uburyo bubiri bwo gukuramo, aho hafi 60% bikurwamo n'umwijima n'ibisigaye bikurwamo n'impyiko. Mu bihe by'imikorere mibi y'impyiko cyangwa umwijima, inzira yindi yo gusohora ishobora kwishyura iyangiritse.

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Amakuru y'inyongera:

Imiterere C29H30N6O6
Isuzuma 99%
Isura Ifu y'umweru kuva kuri beige
Nimero ya CAS 144689-63-4
Gupakira 25KG
Igihe cyo kuruhuka Imyaka 2
Ububiko Bika ahantu hakonje kandi humutse
Icyemezo ISO.

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