Umukandara n'Inzira: Ubufatanye, Ubwumvikane no Gutsinda Ubwuzuzanye
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Ibicuruzwa

Clascoterone CAS:19608-29-8 Umukozi Ukora

Clascoterone ni umuti ugabanya androgen receptor urimo gukorwa nk'amavuta yo mu bwoko bwa cream n'umuti utangwa na Cassiopea (ikigo cy’ubucuruzi cya Cosmo Pharmaceuticals) mu kuvura indwara z'uruhu ziterwa na androgen, harimo alopecia ya androgenetic na acne vulgaris. Nubwo uburyo nyabwo bwo kuvura acne vulgaris butazwi, uyu muti uzwiho guhangana na androgen dihydrotestosterone mu gufatana na androgen receptors mu ngirabuzimafatizo z'umusatsi no mu dusatsi kugira ngo ugabanye ibimenyetso bikenewe kugira ngo acne itere imbere.


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Clascoterone irimo gutegurwa nk'amavuta yo mu bwoko bwa cream na Cassiopea yo kuvura indwara z'uruhu zishingiye kuri androgen. Clascoterone (cortexolone 17α-propionate, CB-03-01) ni umuti mushya w'udusimba twa androgen. Ifatana n'udusimba twa androgen hamwe n'ubukana bwinshi. Mu guhangana na androgens kugira ngo ifatanye na androgens, clascoterone ikora ihagarika uburyo androgen receptor signalling cascades butuma habaho ibiheri, nko kwiyongera kw'uturemangingo twa sebaceous, gukora sebum nyinshi, n'inzira zo kubyimba. Muri Kanama 2020, FDA yemeje clascoterone ku buryo bwo kuvura ibiheri bya mbere (acne vulgaris) ku barwayi b'abagabo n'abagore bafite imyaka 12 kuzamura. Clascoterone irimo gukorwaho ubushakashatsi nk'uburyo bushya bwo kuvura alopecia ya androgenetic.

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Amakuru y'inyongera:

Imiterere C24H34O5
Isuzuma 99%
Isura Ifu y'umweru
Nimero ya CAS 19608-29-8
Gupakira 25KG
Igihe cyo kuruhuka Imyaka 2
Ububiko Bika ahantu hakonje kandi humutse
Icyemezo ISO.

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